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Forskolin (毛喉素) (腺苷酸环化酶激活剂) (RPM0013)

Chemical structure of Forskolin, CAS No.:66575-29-9

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货号: RPM0013
价 格:  300.00
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详细信息

靶点
Forskolin; Coleonol; Colforsin; 毛喉素; 佛司可林; 腺苷酸环化酶激活剂
细胞系
410.5
突变描述
货号###名称### 规格 |||RPM0013###Forskolin (毛喉素) (腺苷酸环化酶激活剂)###1mg/5mg||| - ### 说明书###1 份

Mammalian cells such as human, rat and mouse cells are normally diploid with two alleles.
Homozygote: both alleles were knocked out, mRNA has no signal, no expression of proteins.
Heterozygote: only one allele was knocked out, the mRNA transcript levels was decreased compared to wild type, and the protein expression levels was also lower than that of the wild type.
产品组成
本产品仅用于科研。本产品仅用于科研。该物质可用于多领域研究:干细胞研究中抑 TGF-β 通路促其向特定细胞分化,肿瘤研究中阻肿瘤细胞 EMT 抑转移,还能在纤维化疾病研究中抑成纤维细胞活化并助力药物筛选。
物种
66575-29-9
保存条件
Store at -20℃.store at low temperature,store under nitrogen
Powder: -20°C for 3 years
In solvent: -80°C for 1 year
Shipping with blue ice/Shipping at ambient temperature.keep away from direct sunlight,keep away from moisture,store at low temperature
Powder: -20°C for 3 years
In solvent: -80°C for 1 year
Shipping with blue ice/Shipping at ambient temperature.
运输条件
本产品仅用于科研。细胞信号通路中激活腺苷酸环化酶以探究 cAMP-PKA 通路调控作用,代谢研究中促脂肪分解以助力相关机制研究与药物筛选,还能在药理学实验中验证靶点及评估药物影响。

背景信息

Forskolin (Coleonol) 属于天然产物,是一种腺苷酸环化酶激活剂 (EC50=0.5 μM)。Forskolin 可以增加 cAMP 水平,可以激活 PXR 和 FXR,也可以诱导细胞自噬。Forskolin 对心脏产生正性肌力作用,具有血小板抗凝集和降压作用。

别名
Forskolin; Coleonol; Colforsin; 毛喉素; 佛司可林; 腺苷酸环化酶激活剂